TAK-448 Catalog No.:M30275-C RVD-Hpα also high affinity CB2

RVD-Hpα also high affinity CB2 positive allosteric modulator (Ki=50 nM)

Smiles: CC(C)(C)C(=O)CN1C2=CC=CC=C2N(C[C@@H](NC(=O)NC2=CC(=CC=C2)C(O)=O)C1=O)C1CCCCC1

a novel rho-kinase inhibitor

CAS Number: 2413-38-9

full agonist of α7 nAChRs with EC50 of 18 μM

TAK-448 Catalog No.:M30275-C RVD-Hpα also high affinity CB2TAK 448 (MVT 602) is a potent and full KISS1R agonist with an IC50 of 460 pM and an EC50 of 632 pM. Product information CAS Number: 1234319 68 6 Molecular Weight: 1225. 35 Formula: C58H80N16O14 Chemical Name: N {1 [(1 {[({1 [(1 {[1 carbamoyl 2 (1H indol 3 yl)ethyl]carbamoyl} 4 (N'' methylcarbamimidamido)butyl)carbamoyl] 3 methylbutyl}carbamoyl)amino]carbamoyl} 2 phenylethyl)carbamoyl] 2 hydroxypropyl} 2 ({1 [2 acetamido 3 (4 hydroxyphenyl)propanoyl] 4