MSI-1436 lactate Catalog No.:M33104-C Smiles: CC1C[C@H]2OC(=O)C(=C)[C@H]2[C@H](O)C=1[C@@H](C)CCCO

Smiles: CC1C[C@H]2OC(=O)C(=C)[C@H]2[C@H](O)C=1[C@@H](C)CCCO

PMID: 29926593

CAS Number: 2227548-95-8

In vitro: BAY36-7620 is a potent and selective antagonist at mGlu1receptors and inhibits >60% of mGlu1a receptor constitutive activity (IC50 = 0

GSK-25 has promising oral bioavailability (49% in male Sprague-Dawley rats and 19% in monkey)

MSI-1436 lactate Catalog No.:M33104-C Smiles: CC1C[C@H]2OC(=O)C(=C)[C@H]2[C@H](O)C=1[C@@H](C)CCCOMSI 1436 lactate is a selective, non competitive inhibitor of the enzyme protein tyrosine phosphatase 1B (PTB1B), with an IC50 of 1 M, 200 fold preference over TCPTP (IC50 of 224 M). Product information CAS Number: 1309370 86 2 Molecular Weight: 775. 13 Formula: C40H78N4O8S Chemical Name: 2 hydroxypropanoic acid; {[(3R,6R) 6 [(1R,3aS,3bR,4R,5aR,7S,9aS,9bS,11aR) 7 {[3 ({4 [(3 aminopropyl)amino]butyl}amino)propyl]amino} 4 hydroxy 9a,11a dimethyl