PROTAC ERα Degrader-2 Catalog No.:M7993-2 4-dimethoxyphenethyl)-3-(4-((2-isopropyl-1-methyl-1H-indol-3-yl)sulfonyl)phenoxy)-N-methylpropan-1-amine

4-dimethoxyphenethyl)-3-(4-((2-isopropyl-1-methyl-1H-indol-3-yl)sulfonyl)phenoxy)-N-methylpropan-1-amine

compared with bortezomib

InChi: InChI=1S/C28H28N4O2

It has no activity against CARM1 and Set7/9 methyltransferases

CAS Number: 849217-68-1

PROTAC ERα Degrader-2 Catalog No.:M7993-2 4-dimethoxyphenethyl)-3-(4-((2-isopropyl-1-methyl-1H-indol-3-yl)sulfonyl)phenoxy)-N-methylpropan-1-aminePROTAC ER Degrader 2 comprises a cIAP1 ligand binding group, a linker and an estrogen receptor (ER) binding group. PROTAC ER Degrader 2 is an ER degrader. Maximal ER degradation at 30 M concentration in human mammary tumor MCF7 cells. Degradation inducers based on cIAP1 are called specific and non genetic IAP dependent protein erasers (SNIPERs). Product information CAS Number: 1351169 29 3 Molecular Weight: 763. 96 Formula: C42H61N5O8 Chemical Name: