Glutaminase-IN-1 Size:Contact [email protected] for quotation Smiles: CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3C[C@H](C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C

Smiles: CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3C[C@H](C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C

PubMed PMID: 25450597

Formula: C15H18N4O4S

4 µM) in stress-cultured MEF cells but does not block IRE1α autophosphorylation

GluK2a (15-fold)

Glutaminase-IN-1 Size:Contact [email protected] for quotation Smiles: CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3C[C@H](C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12CGlutaminase IN 1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4 selenadiazole containing kidney type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase IN 1 (CB839 derivative) shows improved cellular uptake and antitumor activity. Product information CAS Number: 2247127 79 1 Molecular Weight: 618. 47 Formula: C26H24F3N7O3Se Chemical Name: 2 (pyridin 2 yl) N {5 [4 (6 {2 [3 (trifluoromethoxy)phenyl]acetamido}pyridazin 3